mercredi 4 avril 2012

Anticancer compounds: summary (march 2012) - Composés anticancéreux: résumé (mars 2012)



Generic Name
Nom générique
Designation
Brand Name
Nom commercial



Abexinostat hydrochloride
PCI-24781 , CRA-024781

Abiraterone acetate
CB7630
Zytiga
Aderbasib
INCB 007839

Afatinib
BIBW2992

Aflibercept
AVE0005, VEGF Trap, VEGF-Trap, NSC 724770
Zaltrap
Agatolimod
PF-3512676

Alemtuzumab

Campath
Alisertib
MLN8237-004

Alvespimycin
KOS-1022

Alvespimycin hydrochloride
BMS-826476

Alvocidib
Flavopiridol, HL-275, HMR-1275, L86-8275, MDL-107826A, NSC-649890

Amatuximab
MORAb-009

Amonafide ???


Amrubicin hydrochloride
SM-5887

Amuvatinib
MP-470, MP470, HPK-56, MP470.HCl

Anamorelin hydrochloride
RC-1291 HCl

Angiopoietin-2
REGN910 SAR307746

Apatinib
YN968D1

Apricoxib
TG01, R-109339, CS-706

Astuprotimut-R
GSK-249553, SB-249553, MAGE-A3 ASCI

Axitinib
AG-13736, AG-013736

Azacitidine

Vidaza
Azacitidine 5’ elaidic ester
CP-4200

Bafetinib
INNO-406, NS-187

Balamapimod
MKI-833

Bardoxolone
RTA 401, CDDO

Bardoxolone methyl
RTA 402, CDDO-Me, NSC 713200

Bavituximab
3G4
Tarvacin
Belagenpumatucel-L

Lucanix
Belinostat
PXD101, NSC 726630

Belotecan hydrochloride
CKD-602

Berubicin hydrochloride
RTA 744, WP744

Bevacizumab

Avastin
Blinatumomab
MEDI-538, MT-103, MT103

Bortezomib

Velcade
Bosutinib
SKI-606 , PF-5208763, SKI-758

Brentuximab vedotin
SGN-35, SGN35, cAC10-vcMMAE
Adcetris
Brivanib
BMS-540215

Brivanib alaninate
BMS-582664

Cabazitaxel
XRP-6258

Cabozantinib (s-malate)
XL184, XL 184, EXEL-7184, BMS 907351

Calaspargase (pegol)
EZN-2285

Camptothecin
IT-101, CRLX101
Cyclosert-CPT
Canertinib
CI-1033

Cantuzumab Ravtansine
huC242-DM4 IMGN242

Carfilzomib
PR-171

Carlumab
CNTO 888

Cediranib (maleate)
AZD2171 (maleate)
Recentin
Cenersen sodium
OL(1)p53, EL625

Cetuximab

Erbitux
Cevipabulin (fumarate or succinate)
TTI-237

Chidamide
HBI-8000, CS055

Cilengitide
EMD 121974, EMD121974

Cixutumumab
IMC-A12

(Yttrium Y90) Clivatuzumab tetraxetan
hPAM4-DOTA ,IMMU-107, 90hY-PAM4

Conatumumab
AMG 655, TRAIL-R2 mAb

Contusugene ladenovec
Ad5CMV-p53, INGN 201

Cordecepin or Cordycepin
BU-01, OVI-123

Cositecan
Karenitecin

BNP1350


Crenolanib (besylate), formerly plarotinib
ARO-002(-26), CP-868,596(-26), CP-868596, ARO-002

Crisantaspase, Erwinia chrysanthemi L-asparaginase

Erwinase, Erwinaze (USA)
Crizotinib
PF-2341066, PF-2,341,066, PF-02341066, PF1066, PF-1066
Xalkori
Crolibulin
EPC2407

Custirsen sodium
OGX-011, ISIS 112989

Cytarabine:daunorubicin
CPX-351

Dabrafenib (mesylate)
GSK-2118436(B)

Dacetuzumab
SGN-40, huS2C6

Dacomitinib
PF-299, PF299804, PF-00299804, PF-299,804, PF00299804

Dalantercept
ACE-041, protéine

Dalotuzumab
MK-0646

Danusertib
PHA-739358

Darinaparsin
ZIO-101

Dasatinib
BMS-354825
Sprycel
Daunorubicin citrate liposome
NSC 82151
DaunoXome
Decitabine

Dacogen
Defibrotide


Deforolimus


Degarelix acetate
FE200486
Firmagon
Delanzomib
CEP18770, CT47098, NPH007098

Demcizumab
OMP-21M18

Denenicokin
L-methionyl(human interleukin-21), IL-21, rIL-21, recombinant human interleukin 21

Denibulin hydrochloride
MN- 029

Desmethyl Erlotinib
OSI-420, CP-473420

Dinaciclib
SCH 727965

Disomotide
MPS-22

Dovitinib
TKI258, CHIR-258

Doxorubicin (zoptarelin)
AN-152, AN 152, ZEN-008, AEZS-108, DOX-LTSL
ThermoDox
Drozitumab
PRO95780, anti-DR5, rhuMAb DR5

Dulanermin
Apo2L/TRAIL, PRO1762, TRAIL/Apo2L, AMG 951
 rhApo2L, RG3639

Edotecarin
PF-804950

Elacytarabine
CP-4055
Elacyt
Elagolix
NBI-56418

Elagolix sodium
NBI-56418 Na

Elesclomol
STA-4783

Elisidepsin
PM02734
Irvalec
Elotuzumab
HuLuc63, PDL063, PDL-063, BMS-901608

Emepepimut-S
L-BLP25, BLP-25 (formerly BP1-7-KLH), EMD531444
Stimuvax
Enavatuzumab
PDL 192

Eniluracil
GW776C85, ADH300004
Cytefuran
Ensituximab
NPC-1C

Entinostat
MS275, SNDX-275, MS-275

Enzastaurin
LY317615

Epetirimod mesylate
851B, S-30563-35-65

Epitinib
HMPL-813

Epratuzumab
Y90 MAb LL2, 90Y-hLL2, IMMU-103, hLL2, hCD22, AMG 412
LymphoCide Y-90
Eribulin mesylate
E7389

Erismodegib
LDE225

Erlotinib

Tarceva
Etaracizumab
Etaratuzumab, MEDI-522
Abegrin
Vitaxin
Everolimus

Afinitor
Falimarev
PANVAC-F, CVAC-301, formerly Panvac-VF

Famitinib


Farletuzumab
MORAb-003

Ficlatuzumab
SCH900105, AV299, AV-299, SCH 900105

Figitumumab
CP-751,871

Flanvotumab
IMC-20DS7

Flumatinib
HHGV678, HH-GV678, HH-GV-678

Folitixorin calcium
ANX-510, CoFactor

Foretinib
GSK1363089G, XL880

Forodesine
BCX-1777, immucillin-H
Fodosine
Fosbretabulin (tromethamine)
combretastatin-A4 phosphate, CA4P
Zybrestat
Fostamatinib
R7935788

Fostamatinib disodium
R788, R-788, R935788 sodium

Fresolimumab
GC1008

Fruquintinib
HMPL-013

Galactomycin
GM-CT-01 (formerly Davanat-1)    
Pro-5FU
Galeterone
TOK-001, VN/124-1, VN/124

Galgenprostucel-L
CG1940
GVAX™ Prostate
Ganetespib
STA-9090

Ganitumab
AMG 479

Gataparsen (sodium)
LY2181308 heptadecasodium salt

Gefitinib

Iressa
Gemcitabine 5'-elaidic acid ester
CP-4126, O-1.01, CO-101

Girentuximab
WX-G250, cG250, anti-G250, cG250

(Iodine I124) girentuximab
124IcG250
Redectane
Givinostat
ITF2357

Glembatumumab vedotin
CR011-vcMMAE, CDX-011

Glufosfamide
D-19575

Golnerminogene pradenovec
ADgv EGR.TNF.11D

Histrelin
Formerly RL0903
Vantas
Icotinib
BPI-2009-H

Icrucumab
IMC-18F1, IMC18F1

Imatinib


Imatinib Mesylate
STI-571, STI571, formerly CGP-57148B
Gleevec (USA, Canada, Israel), Glivec (Europe)
Imetelstat
GRN163L
formerly GRN719

Inalimarev
PANVAC-V, CVAC-301, formerly Panvac-VF

Indibulin
ZIO-301, D-24851

Indisulam
E7070

Ingenol mebutate
PEP-005

Intedanib
BIBF1120

Intetumumab
CNTO-95, CNTO 095, CNTO 95

Iniparib
BSI-201

Interferon-alpha 2b

Biphasix
Iobenguane I 131
MIP-120T, Ultratrace MIBG
Azedra, Ultratrace iobenguane I-131
Ioflubenzamide I131
BA-100, MIP-1145

Ipilimumab
MDX-010, MDX-CTLA-4
Yervoy
Iratumumab
MDX-060

Irosustat
BN83495, STX64, 667 Coumate

Ispinesib
SB-715992

Lapatinib (ditosylate)
572016, GW572016, GW 572016, GSK 572016
Tykerb (USA, EU), Tyverb
Lapuleucel-T
APC8024, BA7072, DN24-02
Neuvenge
Laromustine
VNP40101M, 101M

Lenalidomide
CDC501, CDC-501, CDC-5013, CC5013, CC-5013
Revlimid (formerly Revimid)
Lenvatinib
ER-203492-00

Lenvatinib mesylate
E7080


Lestaurtinib
CEP-701, KT-5555

Leukocyte interleukin injection

Multikine
Leuprolide acetate

Enanton
Lexibulin
CYT997

Linifanib
ABT-869, RG3635

Linsitinib
OSI-906, OSI-906AA

Litronesib
LY2523355, KF89617

Lonafarnib
SCH66336

Lonaprisan
ZK 230211

Lorvotuzumab mertansine
huN901-DM1, BB-10901TAP, BB-10901, IMGN901

Lucatumumab
CHIR-12.12, HCD-122

Marizomib
NPI-0052

Masitinib (mesylate)
Masivet, AB1010

Melphalan

Percutaneous Hepatic Perfusion (PHP)
Milatuzumab
IMMU-115

Mituprotimut-T
Id/KLH

Mocetinostat
MGCD0103

Mocetinostat dihydrobromide


Mogamulizumab
KW-0761, KM8761

Motesanib (diphosphate)
AMG-706, AMG706

Moxetumomab pasudotox
CAT-8015, HA22

Mubritinib
TAK165

Narnatumab
IMC-RON8, IMC RON-8, RON8

Navitoclax dihydrochloride
ABT-263, RG7423, A-855071.0

Necitumumab
IMC-11F8

Neratinib
HKI-272, PF-05208767

Nilotinib
AMN-107
Tasigna
Niraparib
MK-4827

Obatoclax
GX15-070

Obinutuzumab
Ro-5072759, huMAB
GA-101, afutuzumab

Ofatumumab
GSK1841157, HuMax-CD20, 2F2

Olaparib
AZD2281, KU-0059436

Olaratumab
IMC-3G3, IMC3G3

Omacetaxine mepesuccinate
CGX-635, Homoharringtonine

Onartuzumab
PRO143966, MetMAb, RG3638

Orteronel
TAK-700

Oxaliplatin (L-OHP)
1670RB, RP 54780
Eloxatin, Eloxatine, Elplat
Paclitaxel
ANG1005, GRN1005
OncoJan
Palifosfamide
IPM, ZIO-201

Panitumumab

Vectibix
Panobinostat
LBH-589, LBH 589, LBH589, NVP-LBH589, LBH489B, LBH489A

Pazopanib

Votrient
Pegdinetanib
BMS-844203, CT-322, CT322
Adnectin, Angiocept, formerly TriNectin
Pelitinib
EKB-569

Perifosine
KRX-0401, D-21266

Pertuzumab
RG1273, R1273, 2C4, rhuMAb-2C4
Omnitarg
Pictilisib
GDC-0941

Pixantrone dimaleate
BBR 2778
Pixuvir
Pixantrone
Plinabulin
NPI-2358

Plitidepsin
Dehydrodidemnin B

Aplidin R Aplidine
Ponatinib
AP24534




Quarfloxin
CX-3543

Quizartinib
AC220, AC010220

Racotumomab
1E10

Radium223 Chloride

Alpharadin
Ramucirumab
IMC-1121b, IMC 1121B, LY3009806

Ranagengliotucel-T

Glionix
Ranpirnase
Formerly P-30 protein
Onconase
Regorafenib
BAY 73-4506

Resminostat
4SC-201, BYK408740

Retaspimycin hydrochloride
IPI-504, MEDI-561

Ridaforolimus
AP23573, MK-8669

Rigosertib sodium
ON 01910.Na
Estybon
Rindopeptimut
PF-04948568, PF4948568, CDX-110, ALT-110

Rilotumumab
AMG 102

Rituximab

Rituxan
Robatumumab
SCH 717454

Romidepsin

Istodax
Ropidoxuridine
IPdR

Rucaparib
AG-14447

Rucaparib phosphate
AG014699, PF01367338

Ruxolitinib (phosphate)
INC424, INCB018424 (salt)

Sagopilone
DE-03757, ZK 219477, SHY03757, , SH-Y03757A, ZK-219477, ZK-epothilone, BAY86-5302
ZK-EPO
Salirasib
farnesyl thiosalicylic acid

Samalizumab
ALXN6000

Sapacitabine
CYC682, CS-682

Saracatinib
AZD0530

Saracatanib fumarate
AZD0530 fumarate

Saridegib
IPI-926

Seliciclib
R-roscovitine, CYC-202

Selumetinib
AZD6244 , ARRY-142886

Selumetinib sulfate
AZD6244 Hydrogen Sulfate

Semaxinib
SU5416

Sepantronium (bromide)
YM155

Siltuximab
CNTO-328




Sivifene
A-007

Solitomab
MT110

Sorafenib (tosylate)
BAY 43-9006 (BAY 54-9085)
Nexavar
Sotatercept
ACE-011

Squalamine
MSI-1256F
Evizon (ophthalmic)
Sulfatinib
HMPL-012

Sunitinib

Sutent
Talactoferrin alfa, talactoferrin


Talimogene Laherparepvec
OncoVEX GM-CSF, OncoVEXGMCSF, OncoVEXGM-CSF,
JS1 34.5-hGMCSF 47- pA-

Tamoxifen citrate

Soltamox
Tandutinib
MLN0518, MLN518, MLN-518
(formerly CT53518, CT-53518)

Tanespimycin
KOS-953

Tasisulam sodium
LY573636


Tasquinimod
ABR-215050
Tumor Angiogenesis Suppression by Quinolines (TASQ)
Teglanirad chloride
GMX1777, EB1627

Telatinib
BAY 57-9352

Telotristat
LP-778902

Temsirolimus

Torisel
Tenifatecan
SN2310

Teprotumumab
RO4858696-000

Theliatinib
HMPL-309

Tigatuzumab
R-161460, TRA-8, CS-1008

Tipapkinogene sovacivec
TG-4001, TG4001, MVA-HPV-IL2, R3484, RO5217790

Tipifarnib
R115777
Zarnestra
Tivantinib
ARQ-650RP, ARQ 650RP, ARQ 197, ARQ197

Tivozanib
AV-951, AV951
Formerly KRN-951

Tosedostat
CHR-2797

Tozasertib lactate
MK-0457, VX-680

Trametinib
GSK1120212

Trastuzumab

Herceptin
Trastuzumab emtansine
PRO132365, trastuzumab-MCC-DM1 , T-DM1

Trebananib
AMG-386

Tremelimumab (formerly ticilimumab)
CP-675,206, CP-675, CP-675206

Urelumab
BMS-663513

Valrubicin
AD32
Valstar, Valtaxin
Vandetanib
ZD6474, AZD6474, AZD-6474
Caprelsa (formerly Zictifa and Zactima)
Varlitinib
ARRY-334543

Varlitinib tosylate
AR00334543, ARRY-334543, ARRY-543

Vatalanib
PTK787

Veltuzumab
IMMU-106

Veliparib
ABT-888

Veltuzumab
IMMU-106, hA20, hCD20

Vemurafenib
PLX-4032, RG7204, R7204, RO5185426
Zelboraf
Verubulin
MPC-6827, MX-128495
Azixa
Vincristine sulfate liposomes for injection (VSLI)

Marqibo (formerly Onco TCS), Vincristine Optisome
Vinflunine ditartrate
BMS-710485, F-12158
Javlor
Vinorelbine tartrate
ANX-530, formerly SDP-012
Exelbine
Vismodegib
GDC-0449, Cur-691, RG3616
HhAntag
Volasertib
BI6727

Volitinib
HMPL-504

Vorinostat

Zolinza
Vosaroxin
SNS-595, SPC-595, formerly AG-7352, formerly voreloxin

Zalutumumab
HuMax-EGFr, 2F8

Zibotentan
ZD4054





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